產品屬性：
產品名稱 | Tolperisone-d10 (hydrochloride) |
規格 | 500 μg、1 mg |
貨號 | EY-01Y14493 |
Cas No.: 1185160-65-9
別名: N/A
化學名: N/A
分子式: C16H13D10NO.HCl
分子量: 291.9
溶解度:
儲存條件: Store at 2°C to 8°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述：
Tolperisone-d10 is intended for use as an internal standard for the quantification of tolperisone by GC- or LC-MS. Tolperisone is a piperidine that acts as an inhibitor of voltage-gated sodium channels with an IC50 value of 198 μM, for inhibition of peak sodium currents evoked by step depolarizations in dorsal root ganglion (DRG) neurons, in vitro.1 Tolperisone acts as an antispastic agent that attenuates monosynaptic, disynaptic, and polysynaptic reflux response to dorsal root stimulation in vivo. Formulations containing tolperisone are used as analgesics and muscle relaxants.1.Kocsis, P., Farkas, S., Fodor, L., et al.Tolperisone-type drugs inhibit spinal reflexes via blockade of voltage-gated sodium and calcium channelsJ. Pharmacol. Exp. Ther.315(3)1237-1246(2005)
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