產品屬性：
產品名稱 | MT-3014 |
規格 | 100mg、250mg、500mg |
貨號 | EY-01Y15342 |
Cas No.: 1332727-40-8
別名: N/A
化學名: N/A
分子式: C23H25F2N7O
分子量: 453.49
溶解度: Soluble in DMSO
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述：
MT-3014 is a potent, highly selective and brain-penetrated phosphodiesterase 10A (PDE 10A) inhibitor, with IC50s of 0.062 nM and 0.09 nM for human PDE 10A and bovine PDE 10A, respectively[1].
human PDE 10A|0.062 nM (IC50)|bovine PDE 10A|0.09 nM (IC50)
[1]. Koizumi Y, et al. Discovery of a pyrazolo[1,5-a]pyrimidine derivative (MT-3014) as a highly selective PDE10A inhibitor via core structure transformation from the stilbene moiety. Bioorg Med Chem. 2019 Jun 19.
特別提醒公司產品僅供科研使用
