產品屬性:
產品名稱 | LXRβ agonist-2 |
規格 | 100mg、250mg、500mg |
貨號 | EY-01Y15334 |
Cas No.: 1949801-52-8
別名: N/A
化學名: N/A
分子式: C32H31F6N3O7

分子量: 683.59
溶解度: Soluble in DMSO
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述:
LXRβ agonist-2 is a highly potent and β-selective liver X receptor (LXRβ) agonist with EC50 of 7 nM, displays 28.5-fold selectivity over LXRα (EC50=200 nM) and used in the treatment of atherosclerosis[1].EC50: 7 nM (LXRβ), 200 nM (LXRα)[1][1]. Koura M,et al. Discovery of a 2-hydroxyacetophenone derivative as an outstanding linker to enhance potency and β-selectivity of liver X receptor agonist. Bioorg Med Chem. 2016 Aug 15;24(16):3436-46.
特別提醒公司產品僅供科研使用