產品屬性：
產品名稱 | LY-2940094 |
規格 | 10mM*1mL in DMSO、5mg、10mg、25mg、50mg、100mg、200mg、500mg |
貨號 | EY-01Y16907 |
Cas No.: 1307245-86-8
別名: N/A
化學名: N/A
分子式: C22H23ClF2N4O2S
分子量: 480.96
溶解度: DMSO: 41.67 mg/mL (86.64 mM)
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述：
LY-2940094 is a potent, selective and orally available nociceptin receptor (NOP receptor) antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM). LY-2940094 reduces ethanol self-administration in animal models[1].Ki: 0.105 nM (NOP receptor)[1]Kb: 0.166 nM (NOP receptor)[1]LY-2940094 (LY2940094; 3, 10, or 30 mg/kg; 2-3 mL/kg; orally daily; for 4 days) dose-dependently reduces homecage ethanol self-administration in Indiana Alcohol-Preferring (P) and Marchigian Sardinian Alcohol-Preferring (msP) rats, without affecting food/water intake or locomotor activity[1].
特別提醒公司產品僅供科研使用
