產品屬性：
產品名稱 | Stafia-1 |
規格 | 10mM*1 mL in DMSO、5 mg、10 mg、25 mg、50 mg、100 mg |
貨號 | EY-01Y16972 |
Cas No.: N/A
別名: N/A
化學名: N/A
分子式: C24H27O10P
分子量: 506.44
溶解度: DMSO : 250 mg/mL (493.64 mM; Need ultrasonic)
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述：
Stafia-1 is a potent STAT5a inhibitor (K i=10.9 μM, IC50=22.2 μM). Stafia-1 displays high selectivity over STAT5b and other STAT family members[1].Stafia-1 shows at least 9-fold selectivity over STAT5b and higher selectivity against other STAT family members[1].[1]. Natarajan K, et al. Stafia-1: a STAT5a-Selective Inhibitor Developed via Docking-Based Screening of in Silico O-Phosphorylated Fragments. Chemistry. 2020;26(1):148-154.
特別提醒公司產品僅供科研使用
