產品屬性：
產品名稱 | LY3130481 |
規格 | 100mg、250mg、500mg |
貨號 | EY-01Y18033 |
Cas No.: 1610802-47-5
別名: N/A
化學名: N/A
分子式: C19H18N4O3S
分子量: 382.44
溶解度: DMSO: 250 mg/mL (653.70 mM)
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產品描述：
LY3130481 is an AMPA receptor antagonist that is dependent upon transmembrane AMPA receptor regulatory protein (TARP) γ-8, selective inhibits AMPA/TARP γ-8 with an IC50 of 65 nM[1].IC50:65 nM (AMPA/TARP γ-8)[1][1]. Gardinier KM,et al. Discovery of the First α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor Antagonist Dependent upon Transmembrane AMPA Receptor Regulatory Protein (TARP) γ-8. J Med Chem. 2016 May 26;59(10):4753-68.
特別提醒公司產品僅供科研使用
